CYS2, TYR3, ARG5, PEN7-AMIDE

CYS2, TYR3, ARG5, PEN7-AMIDE

CTAP

CAS: 103429-32-9

Molecular Formula: C51H69N13O11S2

CYS2, TYR3, ARG5, PEN7-AMIDE - Names and Identifiers

Name	CTAP
Synonyms	CTAP 7)-disulfide CYS2, TYR3, ARG5, PEN7-AMIDE M.W. 1104.30 C51H69N13O11S2 D-PHE-CYS-TYR-D-TRP-ARG-THR-PEN-THR-NH2 H-D-PHE-CYS-TYR-D-TRP-ARG-THR-PEN-THR-NH2 H-D-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr-NH2(Cys2-Pen7)
CAS	103429-32-9

CYS2, TYR3, ARG5, PEN7-AMIDE - Physico-chemical Properties

Molecular Formula	C51H69N13O11S2
Molar Mass	1104.3
Storage Condition	-20°C

CYS2, TYR3, ARG5, PEN7-AMIDE - Risk and Safety

WGK Germany

3

CYS2, TYR3, ARG5, PEN7-AMIDE - Reference Information

biological activity	CTAP is a potent and highly selective brain osmotic opioid receptor (μ opioid receptor) antagonist (IC50=3.5 nM), which is more than 1200 times selective to δ opioid receptor (IC50=4500 nM) and somatostatin receptor. CTAP can be used in the study of L-dopamine (HY-N0304)-induced dyskinesia (LID).
target	IC50: 3.5 nM (μ opioid receptor)IC50: 4500 nM (δ opioid receptor)

Last Update：2024-04-09 20:49:11

CYS2, TYR3, ARG5, PEN7-AMIDE

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CYS2, TYR3, ARG5, PEN7-AMIDE

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